Molecule Details
InChIKeyKLLYFMFRMYWJND-UHFFFAOYSA-N
Compound Name2,2-dimethyl-6-(pyridin-4-yl)-2,3-dihydrothieno[2,3-d]pyrimidin-4(1H)-one
Canonical SMILESCC1(C)NC(=O)c2cc(-c3ccncc3)sc2N1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.9
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13464 ROCK1 Homo sapiens Human PF25346 PF00069 PF08912 7.0 IC50 ChEMBL;BindingDB
O00311 CDC7 Homo sapiens Human PF00069 6.8 IC50 ChEMBL
Q9UBU7 DBF4 Homo sapiens Human PF07535 6.8 IC50 ChEMBL;BindingDB