Molecule Details
InChIKeyKKZJKNBXDCSEGW-UHFFFAOYSA-N
Compound Name[6-[6-(6-methylpyrazin-2-yl)pyrazolo[4,3-c]pyridin-1-yl]-3,4-dihydro-2H-pyrano[3,2-b]pyridin-3-yl]methanamine
Canonical SMILESCc1cncc(-c2cc3c(cn2)cnn3-c2ccc3c(n2)CC(CN)CO3)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.54
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 9.1 Ki ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 8.8 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 7.7 Ki ChEMBL;BindingDB