Molecule Details
InChIKeyKKMZQQWZVBKDFC-UHFFFAOYSA-N
Compound Name2-Piperazin-1-yl-6-[2-(propan-2-ylamino)-4-pyridinyl]pyridine-4-carboxamide
Canonical SMILESCC(C)Nc1cc(-c2cc(C(N)=O)cc(N3CCNCC3)n2)ccn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.4
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q15139 PRKD1 Homo sapiens Human PF00130 PF00169 PF00069 PF25525 9.0 IC50 ChEMBL;BindingDB
Q13563 PKD2 Homo sapiens Human PF18109 PF08016 PF20519 8.1 IC50 BindingDB
Q9BZL6 PRKD2 Homo sapiens Human PF00130 PF00169 PF00069 PF25525 8.1 IC50 ChEMBL