Molecule Details
InChIKeyKJHBJSSYYMWKLQ-UHFFFAOYSA-N
Compound NameN'-methyl-N'-[[5-[4-(2-methylpropyl)phenyl]-1H-pyrazol-4-yl]methyl]ethane-1,2-diamine
Canonical SMILESCC(C)Cc1ccc(-c2[nH]ncc2CN(C)CCN)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.1
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q99873 PRMT1 Homo sapiens Human PF13649 PF22528 8.3 IC50 ChEMBL;BindingDB
Q96LA8 PRMT6 Homo sapiens Human PF13649 PF22528 8.0 IC50 ChEMBL;BindingDB
Q9NR22 PRMT8 Homo sapiens Human PF06325 PF22528 8.0 IC50 ChEMBL;BindingDB