Molecule Details
InChIKeyKJDDJAPSHCVDDC-UHFFFAOYSA-N
Compound Name4-amino-N-cyclopropyl-8-(3,6-dimethoxypyridazin-4-yl)-7-fluorocinnoline-3-carboxamide
Canonical SMILESCOc1cc(-c2c(F)ccc3c(N)c(C(=O)NC4CC4)nnc23)c(OC)nn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.25
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P18507 GABRG2 Homo sapiens Human PF02931 PF02932 9.2 Ki ChEMBL
P28472 GABRB3 Homo sapiens Human PF02931 PF02932 9.2 Ki ChEMBL
P47869 GABRA2 Homo sapiens Human PF02931 PF02932 9.2 Ki ChEMBL;BindingDB