Molecule Details
InChIKeyKJBINAWDNVGVJU-UHFFFAOYSA-N
Compound Name4-[[[[4-(6-Bromo-13-chloro-4-azatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-ylidene)piperidin-1-yl]-(cyanoamino)methylidene]amino]methyl]piperidine-1-carboxamide
Canonical SMILESN#CN/C(=N/CC1CCN(C(N)=O)CC1)N1CCC(=C2c3ccc(Cl)cc3CCc3cc(Br)cnc32)CC1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.22
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 8.2 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 8.2 IC50 ChEMBL