Molecule Details
InChIKeyKIPSRZQNNGSYJE-UHFFFAOYSA-N
Compound Name2-(3-(tert-butylamino)-2-methylquinoxalin-5-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one
Canonical SMILESCc1nc2cccc(-c3cc4c([nH]3)CCNC4=O)c2nc1NC(C)(C)C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.27
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11309 PIM1 Homo sapiens Human PF00069 9.0 IC50 ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 8.9 IC50 ChEMBL;BindingDB
Q86V86 PIM3 Homo sapiens Human PF00069 7.0 IC50 ChEMBL