Molecule Details
InChIKeyKIBQAHRNVOBWRT-UHFFFAOYSA-N
Compound NamePyrazolo[4,3-h]quinazoline-3-carboxamide, 24
Canonical SMILESCN1CCN(c2cccc(Nc3ncc4c(n3)-c3c(c(C(N)=O)nn3C)CC4)c2)CC1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.26
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P24941 CDK2 Homo sapiens Human PF00069 9.0 pIC50 TTD_MultiTarget
O14965 AURKA Homo sapiens Human PF00069 7.5 IC50 ChEMBL;BindingDB