Molecule Details
| InChIKey | KHVVJKLNKLQLJZ-SFHVURJKSA-N |
|---|---|
| Compound Name | CID 135309104 |
| Canonical SMILES | CN1C(=O)[C@@H](N2CCc3c(nn(Cc4ccccc4)c3Br)C2=O)COc2ccccc21 |
| Clinical Status | Data-mined Candidate |
| Targets (Human+Pathogen) | 288 |
| Pfam Stratification | Cross-Family |
| Avg pChEMBL | 6.01 |
| Source | ChEMBL |
2D Structure
Activity Profile
Target Activities (288)
| Target | Gene | Organism | Category | Pfam | pChEMBL | Type | Source |
|---|---|---|---|---|---|---|---|
| Q13546 | RIPK1 | Homo sapiens | Human | PF00531 PF07714 | 9.1 | IC50 | ChEMBL |
| P14867 | GABRA1 | Homo sapiens | Human | PF02931 PF02932 | 6.5 | Ki | ChEMBL |
| O00238 | BMPR1B | Homo sapiens | Human | PF01064 PF07714 PF08515 | 6.0 | IC50 | ChEMBL |
| O00311 | CDC7 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| O00329 | PIK3CD | Homo sapiens | Human | PF00454 PF00792 PF02192 PF00794 PF00613 | 6.0 | IC50 | ChEMBL |
| O00444 | PLK4 | Homo sapiens | Human | PF00069 PF18190 PF18409 | 6.0 | IC50 | ChEMBL |
| O14578 | CIT | Homo sapiens | Human | PF00780 PF00169 PF00069 PF00433 | 6.0 | IC50 | ChEMBL |
| O14757 | CHEK1 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| O14920 | IKBKB | Homo sapiens | Human | PF18397 PF12179 PF00069 | 6.0 | IC50 | ChEMBL |
| O14936 | CASK | Homo sapiens | Human | PF00625 PF02828 PF00595 PF00069 PF07653 | 6.0 | IC50 | ChEMBL |
| O14965 | AURKA | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| O14976 | GAK | Homo sapiens | Human | PF00069 PF10409 | 6.0 | IC50 | ChEMBL |
| O15021 | MAST4 | Homo sapiens | Human | PF08926 PF17820 PF00069 | 6.0 | IC50 | ChEMBL |
| O15111 | CHUK | Homo sapiens | Human | PF18397 PF12179 PF00069 | 6.0 | IC50 | ChEMBL |
| O15146 | MUSK | Homo sapiens | Human | PF01392 PF07679 PF13927 PF07714 | 6.0 | IC50 | ChEMBL |
| O15264 | MAPK13 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| O15530 | PDPK1 | Homo sapiens | Human | PF14593 PF00069 | 6.0 | IC50 | ChEMBL |
| O43283 | MAP3K13 | Homo sapiens | Human | PF07714 | 6.0 | IC50 | ChEMBL |
| O43293 | DAPK3 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| O43318 | MAP3K7 | Homo sapiens | Human | PF07714 | 6.0 | IC50 | ChEMBL |
| O43353 | RIPK2 | Homo sapiens | Human | PF00619 PF07714 | 6.0 | IC50 | ChEMBL |
| O43683 | BUB1 | Homo sapiens | Human | PF08311 PF00069 | 6.0 | IC50 | ChEMBL |
| O60285 | NUAK1 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| O60307 | MAST3 | Homo sapiens | Human | PF08926 PF17820 PF00069 | 6.0 | IC50 | ChEMBL |
| O60885 | BRD4 | Homo sapiens | Human | PF17035 PF17105 PF00439 | 6.0 | IC50 | ChEMBL |
| O75116 | ROCK2 | Homo sapiens | Human | PF25346 PF00069 PF08912 | 6.0 | IC50 | ChEMBL |
| O75385 | ULK1 | Homo sapiens | Human | PF12063 PF21127 PF00069 | 6.0 | IC50 | ChEMBL |
| O75460 | ERN1 | Homo sapiens | Human | PF00069 PF06479 | 6.0 | IC50 | ChEMBL |
| O75582 | RPS6KA5 | Homo sapiens | Human | PF00069 PF00433 | 6.0 | IC50 | ChEMBL |
| O75676 | RPS6KA4 | Homo sapiens | Human | PF00069 PF00433 | 6.0 | IC50 | ChEMBL |
| O94806 | PRKD3 | Homo sapiens | Human | PF00130 PF00169 PF00069 PF25525 | 6.0 | IC50 | ChEMBL |
| O94921 | CDK14 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| O95747 | OXSR1 | Homo sapiens | Human | PF12202 PF00069 | 6.0 | IC50 | ChEMBL |
| O95819 | MAP4K4 | Homo sapiens | Human | PF00780 PF00069 | 6.0 | IC50 | ChEMBL |
| O95835 | LATS1 | Homo sapiens | Human | PF00069 PF00433 PF00627 | 6.0 | IC50 | ChEMBL |
| O96013 | PAK4 | Homo sapiens | Human | PF00786 PF00069 | 6.0 | IC50 | ChEMBL |
| O96017 | CHEK2 | Homo sapiens | Human | PF00498 PF00069 | 6.0 | IC50 | ChEMBL |
| P00519 | ABL1 | Homo sapiens | Human | PF08919 PF07714 PF00017 PF00018 | 6.0 | IC50 | ChEMBL |
| P00533 | EGFR | Homo sapiens | Human | PF00757 PF14843 PF07714 PF01030 PF21314 | 6.0 | IC50 | ChEMBL |
| P04629 | NTRK1 | Homo sapiens | Human | PF13855 PF16920 PF07714 PF18613 | 6.0 | IC50 | ChEMBL |
| P05771 | PRKCB | Homo sapiens | Human | PF00130 PF00168 PF00069 PF00433 | 6.0 | IC50 | ChEMBL |
| P06213 | INSR | Homo sapiens | Human | PF00757 PF17870 PF07714 PF01030 | 6.0 | IC50 | ChEMBL |
| P06239 | LCK | Homo sapiens | Human | PF07714 PF00017 PF00018 | 6.0 | IC50 | ChEMBL |
| P06493 | CDK1 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| P07332 | FES | Homo sapiens | Human | PF00611 PF07714 PF00017 | 6.0 | IC50 | ChEMBL |
| P07333 | CSF1R | Homo sapiens | Human | PF00047 PF25305 PF07714 | 6.0 | IC50 | ChEMBL |
| P08069 | IGF1R | Homo sapiens | Human | PF00757 PF07714 PF01030 | 6.0 | IC50 | ChEMBL |
| P08631 | HCK | Homo sapiens | Human | PF07714 PF00017 PF00018 | 6.0 | IC50 | ChEMBL |
| P08922 | ROS1 | Homo sapiens | Human | PF00041 PF07714 | 6.0 | IC50 | ChEMBL |
| P09619 | PDGFRB | Homo sapiens | Human | PF00047 PF13927 PF25305 PF07714 | 6.0 | IC50 | ChEMBL |
| P09769 | FGR | Homo sapiens | Human | PF07714 PF00017 PF00018 | 6.0 | IC50 | ChEMBL |
| P0C1S8 | WEE2 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| P0C264 | SBK3 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| P10721 | KIT | Homo sapiens | Human | PF00047 PF07714 | 6.0 | IC50 | ChEMBL |
| P11309 | PIM1 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| P11801 | PSKH1 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| P11802 | CDK4 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| P14616 | INSRR | Homo sapiens | Human | PF00041 PF00757 PF07714 PF01030 | 6.0 | IC50 | ChEMBL |
| P15056 | BRAF | Homo sapiens | Human | PF00130 PF07714 PF02196 | 6.0 | IC50 | ChEMBL |
| P16591 | FER | Homo sapiens | Human | PF00611 PF07714 PF00017 | 6.0 | IC50 | ChEMBL |
| P17252 | PRKCA | Homo sapiens | Human | PF00130 PF00168 PF00069 PF00433 | 6.0 | IC50 | ChEMBL |
| P17612 | PRKACA | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| P17948 | FLT1 | Homo sapiens | Human | PF07679 PF00047 PF13927 PF22971 PF07714 PF21339 PF17988 PF22854 | 6.0 | IC50 | ChEMBL |
| P19525 | EIF2AK2 | Homo sapiens | Human | PF00035 PF00069 | 6.0 | IC50 | ChEMBL |
| P19784 | CSNK2A2 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| P21709 | EPHA1 | Homo sapiens | Human | PF14575 PF25599 PF01404 PF07699 PF00041 PF07714 PF00536 | 6.0 | IC50 | ChEMBL |
| P22455 | FGFR4 | Homo sapiens | Human | PF07679 PF13927 PF07714 | 6.0 | IC50 | ChEMBL |
| P22607 | FGFR3 | Homo sapiens | Human | PF21165 PF07679 PF13927 PF07714 | 6.0 | IC50 | ChEMBL |
| P22612 | PRKACG | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| P22694 | PRKACB | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| P23443 | RPS6KB1 | Homo sapiens | Human | PF00069 PF00433 | 6.0 | IC50 | ChEMBL |
| P24723 | PRKCH | Homo sapiens | Human | PF00130 PF00168 PF00069 PF00433 | 6.0 | IC50 | ChEMBL |
| P24941 | CDK2 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| P25098 | GRK2 | Homo sapiens | Human | PF00169 PF00069 PF00615 | 6.0 | IC50 | ChEMBL |
| P27037 | ACVR2A | Homo sapiens | Human | PF01064 PF00069 | 6.0 | IC50 | ChEMBL |
| P27361 | MAPK3 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| P27448 | MARK3 | Homo sapiens | Human | PF02149 PF00069 PF00627 | 6.0 | IC50 | ChEMBL |
| P28482 | MAPK1 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| P29320 | EPHA3 | Homo sapiens | Human | PF14575 PF25599 PF01404 PF07699 PF00041 PF07714 PF07647 | 6.0 | IC50 | ChEMBL |
| P29322 | EPHA8 | Homo sapiens | Human | PF14575 PF25599 PF01404 PF00041 PF07714 PF00536 | 6.0 | IC50 | ChEMBL |
| P29323 | EPHB2 | Homo sapiens | Human | PF14575 PF25599 PF01404 PF07699 PF00041 PF07714 PF00536 | 6.0 | IC50 | ChEMBL |
| P29376 | LTK | Homo sapiens | Human | PF12810 PF07714 | 6.0 | IC50 | ChEMBL |
| P29597 | TYK2 | Homo sapiens | Human | PF18379 PF18377 PF17887 PF07714 PF21990 | 6.0 | IC50 | ChEMBL |
| P30291 | WEE1 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| P30530 | AXL | Homo sapiens | Human | PF00041 PF13927 PF07714 | 6.0 | IC50 | ChEMBL |
| P31152 | MAPK4 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| P31751 | AKT2 | Homo sapiens | Human | PF00169 PF00069 PF00433 | 6.0 | IC50 | ChEMBL |
| P32298 | GRK4 | Homo sapiens | Human | PF00069 PF00615 | 6.0 | IC50 | ChEMBL |
| P34947 | GRK5 | Homo sapiens | Human | PF00069 PF00615 | 6.0 | IC50 | ChEMBL |
| P35557 | GCK | Homo sapiens | Human | PF00349 PF03727 | 6.0 | IC50 | ChEMBL |
| P35626 | GRK3 | Homo sapiens | Human | PF00169 PF00069 PF00615 | 6.0 | IC50 | ChEMBL |
| P35916 | FLT4 | Homo sapiens | Human | PF07679 PF13927 PF22971 PF07714 PF21339 PF17988 PF22854 | 6.0 | IC50 | ChEMBL |
| P35968 | KDR | Homo sapiens | Human | PF07679 PF00047 PF13895 PF22971 PF07714 PF21339 PF17988 PF22854 | 6.0 | IC50 | ChEMBL |
| P36888 | FLT3 | Homo sapiens | Human | PF00047 PF07714 | 6.0 | IC50 | ChEMBL |
| P36894 | BMPR1A | Homo sapiens | Human | PF01064 PF07714 PF08515 | 6.0 | IC50 | ChEMBL |
| P36897 | TGFBR1 | Homo sapiens | Human | PF01064 PF00069 PF08515 | 6.0 | IC50 | ChEMBL |
| P37023 | ACVRL1 | Homo sapiens | Human | PF07714 PF08515 | 6.0 | IC50 | ChEMBL |
| P37173 | TGFBR2 | Homo sapiens | Human | PF08917 PF07714 | 6.0 | IC50 | ChEMBL |
| P41240 | CSK | Homo sapiens | Human | PF07714 PF00017 PF00018 | 6.0 | IC50 | ChEMBL |
| P41743 | PRKCI | Homo sapiens | Human | PF00130 PF00564 PF00069 PF00433 | 6.0 | IC50 | ChEMBL |
| P42336 | PIK3CA | Homo sapiens | Human | PF00454 PF00792 PF02192 PF00794 PF00613 | 6.0 | IC50 | ChEMBL |
| P42338 | PIK3CB | Homo sapiens | Human | PF00454 PF00792 PF02192 PF00794 PF00613 | 6.0 | IC50 | ChEMBL |
| P42680 | TEC | Homo sapiens | Human | PF00779 PF00169 PF07714 PF00017 PF00018 | 6.0 | IC50 | ChEMBL |
| P42681 | TXK | Homo sapiens | Human | PF07714 PF00017 PF00018 | 6.0 | IC50 | ChEMBL |
| P42684 | ABL2 | Homo sapiens | Human | PF08919 PF07714 PF00017 PF00018 | 6.0 | IC50 | ChEMBL |
| P42685 | FRK | Homo sapiens | Human | PF07714 PF00017 PF00018 | 6.0 | IC50 | ChEMBL |
| P43250 | GRK6 | Homo sapiens | Human | PF00069 PF00615 | 6.0 | IC50 | ChEMBL |
| P43405 | SYK | Homo sapiens | Human | PF07714 PF00017 | 6.0 | IC50 | ChEMBL |
| P45983 | MAPK8 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| P45984 | MAPK9 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| P48729 | CSNK1A1 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| P48730 | CSNK1D | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| P49137 | MAPKAPK2 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| P49336 | CDK8 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| P49674 | CSNK1E | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| P49759 | CLK1 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| P49760 | CLK2 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| P49761 | CLK3 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| P49841 | GSK3B | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| P50613 | CDK7 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| P50750 | CDK9 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| P51451 | BLK | Homo sapiens | Human | PF07714 PF00017 PF00018 | 6.0 | IC50 | ChEMBL |
| P51813 | BMX | Homo sapiens | Human | PF00779 PF00169 PF07714 PF00017 | 6.0 | IC50 | ChEMBL |
| P51817 | PRKX | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| P51955 | NEK2 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| P51956 | NEK3 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| P52333 | JAK3 | Homo sapiens | Human | PF18379 PF18377 PF17887 PF07714 PF21990 | 6.0 | IC50 | ChEMBL |
| P52564 | MAP2K6 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| P53350 | PLK1 | Homo sapiens | Human | PF00069 PF00659 | 6.0 | IC50 | ChEMBL |
| P53355 | DAPK1 | Homo sapiens | Human | PF00023 PF12796 PF13637 PF00531 PF00069 | 6.0 | IC50 | ChEMBL |
| P53667 | LIMK1 | Homo sapiens | Human | PF00412 PF00595 PF07714 | 6.0 | IC50 | ChEMBL |
| P53671 | LIMK2 | Homo sapiens | Human | PF00412 PF00595 PF07714 | 6.0 | IC50 | ChEMBL |
| P53778 | MAPK12 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| P53779 | MAPK10 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| P54646 | PRKAA2 | Homo sapiens | Human | PF16579 PF21147 PF00069 | 6.0 | IC50 | ChEMBL |
| P54753 | EPHB3 | Homo sapiens | Human | PF14575 PF25599 PF01404 PF07699 PF00041 PF07714 PF00536 | 6.0 | IC50 | ChEMBL |
| P54756 | EPHA5 | Homo sapiens | Human | PF14575 PF25599 PF01404 PF00041 PF07714 PF00536 | 6.0 | IC50 | ChEMBL |
| P54760 | EPHB4 | Homo sapiens | Human | PF14575 PF25599 PF01404 PF07699 PF00041 PF07714 PF00536 | 6.0 | IC50 | ChEMBL |
| P54762 | EPHB1 | Homo sapiens | Human | PF14575 PF25599 PF01404 PF00041 PF07714 PF00536 | 6.0 | IC50 | ChEMBL |
| P54764 | EPHA4 | Homo sapiens | Human | PF14575 PF25599 PF01404 PF00041 PF07714 PF07647 | 6.0 | IC50 | ChEMBL |
| P57058 | HUNK | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| P57059 | SIK1 | Homo sapiens | Human | PF00069 PF23312 | 6.0 | IC50 | ChEMBL |
| P68400 | CSNK2A1 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| P78362 | SRPK2 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| P78368 | CSNK1G2 | Homo sapiens | Human | PF12605 PF00069 | 6.0 | IC50 | ChEMBL |
| P80192 | MAP3K9 | Homo sapiens | Human | PF07714 PF14604 | 6.0 | IC50 | ChEMBL |
| Q00526 | CDK3 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q00534 | CDK6 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q00535 | CDK5 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q00536 | CDK16 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q00537 | CDK17 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q02156 | PRKCE | Homo sapiens | Human | PF00130 PF00168 PF00069 PF00433 | 6.0 | IC50 | ChEMBL |
| Q02750 | MAP2K1 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q04759 | PRKCQ | Homo sapiens | Human | PF00130 PF21494 PF00069 PF00433 | 6.0 | IC50 | ChEMBL |
| Q04771 | ACVR1 | Homo sapiens | Human | PF01064 PF07714 PF08515 | 6.0 | IC50 | ChEMBL |
| Q05513 | PRKCZ | Homo sapiens | Human | PF00130 PF00564 PF00069 PF00433 | 6.0 | IC50 | ChEMBL |
| Q05655 | PRKCD | Homo sapiens | Human | PF00130 PF21494 PF00069 PF00433 | 6.0 | IC50 | ChEMBL |
| Q06187 | BTK | Homo sapiens | Human | PF00779 PF00169 PF07714 PF00017 PF00018 | 6.0 | IC50 | ChEMBL |
| Q07002 | CDK18 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q07912 | TNK2 | Homo sapiens | Human | PF09027 PF11555 PF07714 PF22931 PF14604 | 6.0 | IC50 | ChEMBL |
| Q08881 | ITK | Homo sapiens | Human | PF00779 PF00169 PF07714 PF00017 PF00018 | 6.0 | IC50 | ChEMBL |
| Q09013 | DMPK | Homo sapiens | Human | PF08826 PF00069 | 6.0 | IC50 | ChEMBL |
| Q12852 | MAP3K12 | Homo sapiens | Human | PF07714 | 6.0 | IC50 | ChEMBL |
| Q12866 | MERTK | Homo sapiens | Human | PF00041 PF00047 PF13927 PF07714 | 6.0 | IC50 | ChEMBL |
| Q13043 | STK4 | Homo sapiens | Human | PF11629 PF00069 | 6.0 | IC50 | ChEMBL |
| Q13131 | PRKAA1 | Homo sapiens | Human | PF16579 PF21147 PF00069 | 6.0 | IC50 | ChEMBL |
| Q13188 | STK3 | Homo sapiens | Human | PF11629 PF00069 | 6.0 | IC50 | ChEMBL |
| Q13237 | PRKG2 | Homo sapiens | Human | PF00027 PF00069 | 6.0 | IC50 | ChEMBL |
| Q13464 | ROCK1 | Homo sapiens | Human | PF25346 PF00069 PF08912 | 6.0 | IC50 | ChEMBL |
| Q13470 | TNK1 | Homo sapiens | Human | PF07714 PF22931 | 6.0 | IC50 | ChEMBL |
| Q13627 | DYRK1A | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q13873 | BMPR2 | Homo sapiens | Human | PF01064 PF00069 | 6.0 | IC50 | ChEMBL |
| Q13882 | PTK6 | Homo sapiens | Human | PF07714 PF00017 PF00018 | 6.0 | IC50 | ChEMBL |
| Q14004 | CDK13 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q14164 | IKBKE | Homo sapiens | Human | PF00069 PF18394 PF18396 | 6.0 | IC50 | ChEMBL |
| Q14289 | PTK2B | Homo sapiens | Human | PF21477 PF00373 PF18038 PF03623 PF07714 | 6.0 | IC50 | ChEMBL |
| Q14680 | MELK | Homo sapiens | Human | PF02149 PF00069 PF21594 | 6.0 | IC50 | ChEMBL |
| Q15139 | PRKD1 | Homo sapiens | Human | PF00130 PF00169 PF00069 PF25525 | 6.0 | IC50 | ChEMBL |
| Q15303 | ERBB4 | Homo sapiens | Human | PF00757 PF14843 PF07714 PF01030 PF21314 | 6.0 | IC50 | ChEMBL |
| Q15349 | RPS6KA2 | Homo sapiens | Human | PF00069 PF00433 | 6.0 | IC50 | ChEMBL |
| Q15375 | EPHA7 | Homo sapiens | Human | PF14575 PF25599 PF01404 PF07699 PF00041 PF07714 PF00536 | 6.0 | IC50 | ChEMBL |
| Q15418 | RPS6KA1 | Homo sapiens | Human | PF00069 PF00433 | 6.0 | IC50 | ChEMBL |
| Q15746 | MYLK | Homo sapiens | Human | PF16620 PF00041 PF07679 PF00069 | 6.0 | IC50 | ChEMBL |
| Q15759 | MAPK11 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q15835 | GRK1 | Homo sapiens | Human | PF00069 PF00615 | 6.0 | IC50 | ChEMBL |
| Q16288 | NTRK3 | Homo sapiens | Human | PF07679 PF00047 PF13855 PF16920 PF01462 PF07714 | 6.0 | IC50 | ChEMBL |
| Q16512 | PKN1 | Homo sapiens | Human | PF02185 PF00069 PF00433 | 6.0 | IC50 | ChEMBL |
| Q16513 | PKN2 | Homo sapiens | Human | PF02185 PF00069 PF00433 | 6.0 | IC50 | ChEMBL |
| Q16539 | MAPK14 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q16566 | CAMK4 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q16584 | MAP3K11 | Homo sapiens | Human | PF07714 PF14604 | 6.0 | IC50 | ChEMBL |
| Q16659 | MAPK6 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q16816 | PHKG1 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q32MK0 | MYLK3 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q52WX2 | SBK1 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q58F21 | BRDT | Homo sapiens | Human | PF17035 PF17105 PF00439 | 6.0 | IC50 | ChEMBL |
| Q59H18 | TNNI3K | Homo sapiens | Human | PF12796 PF07714 | 6.0 | IC50 | ChEMBL |
| Q5VT25 | CDC42BPA | Homo sapiens | Human | PF00130 PF00780 PF08826 PF15796 PF25346 PF00069 PF00433 | 6.0 | IC50 | ChEMBL |
| Q6P2M8 | PNCK | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q6P3R8 | NEK5 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q6PHR2 | ULK3 | Homo sapiens | Human | PF04212 PF00069 | 6.0 | IC50 | ChEMBL |
| Q7KZI7 | MARK2 | Homo sapiens | Human | PF02149 PF00069 PF00627 | 6.0 | IC50 | ChEMBL |
| Q7RTN6 | STRADA | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q86SG6 | NEK8 | Homo sapiens | Human | PF00069 PF25390 | 6.0 | IC50 | ChEMBL |
| Q86UX6 | STK32C | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q86V86 | PIM3 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q86Y07 | VRK2 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q86YV6 | MYLK4 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q86Z02 | HIPK1 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q8IW41 | MAPKAPK5 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q8IYT8 | ULK2 | Homo sapiens | Human | PF12063 PF21127 PF00069 | 6.0 | IC50 | ChEMBL |
| Q8N752 | CSNK1A1L | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q8NB16 | MLKL | Homo sapiens | Human | PF22215 PF07714 | 6.0 | IC50 | ChEMBL |
| Q8NE63 | HIPK4 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q8NFD2 | ANKK1 | Homo sapiens | Human | PF00023 PF12796 PF13637 PF07714 | 6.0 | IC50 | ChEMBL |
| Q8NG66 | NEK11 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q8TD08 | MAPK15 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q8TD19 | NEK9 | Homo sapiens | Human | PF00069 PF25390 | 6.0 | IC50 | ChEMBL |
| Q8TDC3 | BRSK1 | Homo sapiens | Human | PF21122 PF00069 PF21115 | 6.0 | IC50 | ChEMBL |
| Q8WU08 | STK32A | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q8WXR4 | MYO3B | Homo sapiens | Human | PF00612 PF00063 PF00069 | 6.0 | IC50 | ChEMBL |
| Q92630 | DYRK2 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q92918 | MAP4K1 | Homo sapiens | Human | PF00780 PF00069 | 6.0 | IC50 | ChEMBL |
| Q96BR1 | SGK3 | Homo sapiens | Human | PF00069 PF00433 PF00787 | 6.0 | IC50 | ChEMBL |
| Q96GD4 | AURKB | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q96GX5 | MASTL | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q96NX5 | CAMK1G | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q96PY6 | NEK1 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q96RG2 | PASK | Homo sapiens | Human | PF13426 PF00069 | 6.0 | IC50 | ChEMBL |
| Q96S53 | TESK2 | Homo sapiens | Human | PF07714 | 6.0 | IC50 | ChEMBL |
| Q96SB4 | SRPK1 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q99558 | MAP3K14 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q99683 | MAP3K5 | Homo sapiens | Human | PF19039 PF20309 PF20302 PF13281 PF00069 | 6.0 | IC50 | ChEMBL |
| Q99986 | VRK1 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q9BQI3 | EIF2AK1 | Homo sapiens | Human | PF22949 PF00069 | 6.0 | IC50 | ChEMBL |
| Q9BVS4 | RIOK2 | Homo sapiens | Human | PF01163 PF09202 | 6.0 | IC50 | ChEMBL |
| Q9BXA7 | TSSK1B | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q9BXM7 | PINK1 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q9BYT3 | STK33 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q9BZL6 | PRKD2 | Homo sapiens | Human | PF00130 PF00169 PF00069 PF25525 | 6.0 | IC50 | ChEMBL |
| Q9C098 | DCLK3 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q9H093 | NUAK2 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q9H0K1 | SIK2 | Homo sapiens | Human | PF00069 PF23312 | 6.0 | IC50 | ChEMBL |
| Q9H1R3 | MYLK2 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q9H2G2 | SLK | Homo sapiens | Human | PF00069 PF12474 | 6.0 | IC50 | ChEMBL |
| Q9H2K8 | TAOK3 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q9H2X6 | HIPK2 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q9H3Y6 | SRMS | Homo sapiens | Human | PF07714 PF00017 | 6.0 | IC50 | ChEMBL |
| Q9H4B4 | PLK3 | Homo sapiens | Human | PF00069 PF00659 | 6.0 | IC50 | ChEMBL |
| Q9HAZ1 | CLK4 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q9HBY8 | SGK2 | Homo sapiens | Human | PF00069 PF00433 | 6.0 | IC50 | ChEMBL |
| Q9HCP0 | CSNK1G1 | Homo sapiens | Human | PF12605 PF00069 | 6.0 | IC50 | ChEMBL |
| Q9NQU5 | PAK6 | Homo sapiens | Human | PF00786 PF00069 | 6.0 | IC50 | ChEMBL |
| Q9NR20 | DYRK4 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q9NRM7 | LATS2 | Homo sapiens | Human | PF00069 PF00433 | 6.0 | IC50 | ChEMBL |
| Q9NSY1 | BMP2K | Homo sapiens | Human | PF15282 PF00069 | 6.0 | IC50 | ChEMBL |
| Q9NWZ3 | IRAK4 | Homo sapiens | Human | PF07714 | 6.0 | IC50 | ChEMBL |
| Q9NY57 | STK32B | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q9NYL2 | MAP3K20 | Homo sapiens | Human | PF07714 PF07647 | 6.0 | IC50 | ChEMBL |
| Q9NYV4 | CDK12 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q9NZJ5 | EIF2AK3 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q9P0L2 | MARK1 | Homo sapiens | Human | PF02149 PF00069 PF00627 | 6.0 | IC50 | ChEMBL |
| Q9P1W9 | PIM2 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q9P286 | PAK5 | Homo sapiens | Human | PF00786 PF00069 | 6.0 | IC50 | ChEMBL |
| Q9P289 | STK26 | Homo sapiens | Human | PF20929 PF00069 | 6.0 | IC50 | ChEMBL |
| Q9P2K8 | EIF2AK4 | Homo sapiens | Human | PF12745 PF00069 PF05773 PF13393 | 6.0 | IC50 | ChEMBL |
| Q9UBE8 | NLK | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q9UEW8 | STK39 | Homo sapiens | Human | PF12202 PF00069 | 6.0 | IC50 | ChEMBL |
| Q9UF33 | EPHA6 | Homo sapiens | Human | PF14575 PF25599 PF01404 PF07699 PF00041 PF07714 PF00536 | 6.0 | IC50 | ChEMBL |
| Q9UHD2 | TBK1 | Homo sapiens | Human | PF00069 PF18394 PF18396 | 6.0 | IC50 | ChEMBL |
| Q9UIK4 | DAPK2 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q9UK32 | RPS6KA6 | Homo sapiens | Human | PF00069 PF00433 | 6.0 | IC50 | ChEMBL |
| Q9UKE5 | TNIK | Homo sapiens | Human | PF00780 PF00069 | 6.0 | IC50 | ChEMBL |
| Q9UKI8 | TLK1 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q9UL54 | TAOK2 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q9UM73 | ALK | Homo sapiens | Human | PF12810 PF00629 PF07714 | 6.0 | IC50 | ChEMBL |
| Q9UPE1 | SRPK3 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q9UPZ9 | CILK1 | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q9UQ88 | CDK11A | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q9Y243 | AKT3 | Homo sapiens | Human | PF00169 PF00069 PF00433 | 6.0 | IC50 | ChEMBL |
| Q9Y2H9 | MAST1 | Homo sapiens | Human | PF08926 PF17820 PF00069 | 6.0 | IC50 | ChEMBL |
| Q9Y2K2 | SIK3 | Homo sapiens | Human | PF00069 PF23312 | 6.0 | IC50 | ChEMBL |
| Q9Y463 | DYRK1B | Homo sapiens | Human | PF00069 | 6.0 | IC50 | ChEMBL |
| Q9Y4K4 | MAP4K5 | Homo sapiens | Human | PF00780 PF00069 | 6.0 | IC50 | ChEMBL |
| Q9Y572 | RIPK3 | Homo sapiens | Human | PF00069 PF12721 | 6.0 | IC50 | ChEMBL |
| Q9Y616 | IRAK3 | Homo sapiens | Human | PF00531 PF00069 | 6.0 | IC50 | ChEMBL |
| Q9Y6E0 | STK24 | Homo sapiens | Human | PF20929 PF00069 | 6.0 | IC50 | ChEMBL |
| Q9Y6M4 | CSNK1G3 | Homo sapiens | Human | PF12605 PF00069 | 6.0 | IC50 | ChEMBL |