Molecule Details
InChIKeyKHNMKPXPIOAOHB-WPWMEQJKSA-N
Compound Name8-hydroxy-5-[4-[4-[3-[(E)-hydroxyiminomethyl]pyrazolo[1,5-a]pyridin-5-yl]oxybutyl]piperazin-1-yl]-1H-quinolin-2-one
Canonical SMILESO=c1ccc2c(N3CCN(CCCCOc4ccn5ncc(/C=N/O)c5c4)CC3)ccc(O)c2[nH]1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.46
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P14416 DRD2 Homo sapiens Human PF00001 8.8 Ki ChEMBL;BindingDB
P35462 DRD3 Homo sapiens Human PF00001 8.6 Ki ChEMBL;BindingDB
P21917 DRD4 Homo sapiens Human PF00001 8.0 Ki ChEMBL;BindingDB