Molecule Details
InChIKeyKHIURKSPHCFKCV-XCACKJMTSA-N
Canonical SMILESCCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5C[C@H]6CC[C@@H](C5)N6)nc(OC[C@@H]5CCCN5CCCCOCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)c5ccc(-c6scnc6C)cc5)C(C)(C)C)nc4c3F)c12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.52
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P01116 KRAS Homo sapiens Human PF00071 7.5 IC50 ChEMBL
P40337 VHL Homo sapiens Human PF01847 PF17211 7.5 IC50 ChEMBL