Molecule Details
InChIKeyKHGXQGMNQMAHKJ-QSAKORRRSA-N
Compound Name1-[(1-Carboxy-3-methyl-butylcarbamoyl)-(2-{3-methyl-2-[3-methyl-2-(3-phenyl-propionylamino)-butyrylamino]-butyrylamino}-4-oxo-4-pyrrolidin-1-yl-butyrylamino)-methyl]-cyclopentanecarboxylic acid
Canonical SMILESCC(C)C[C@H](NC(=O)[C@@H](NC(=O)[C@H](CC(=O)N1CCCC1)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)CCc1ccccc1)C(C)C)C(C)C)C1(C(=O)O)CCCC1)C(=O)O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.48
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P23921 RRM1 Homo sapiens Human PF03477 PF02867 PF00317 9.0 IC50 ChEMBL;BindingDB
P31350 RRM2 Homo sapiens Human PF00268 8.2 IC50 ChEMBL
Q7LG56 RRM2B Homo sapiens Human PF00268 8.2 IC50 ChEMBL