Molecule Details
InChIKeyKFYKXJYCULQGMU-PTNGSMBKSA-N
Compound Name(Z)-3-(2-{[5-(N,N-Dimethylsulfamoyl)-2-oxoindolin-3-ylidene]-methyl}-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)propanoic Acid
Canonical SMILESCN(C)S(=O)(=O)c1ccc2c(c1)/C(=C/c1[nH]c3c(c1CCC(=O)O)C(=O)CCC3)C(=O)N2
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.68
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O14965 AURKA Homo sapiens Human PF00069 7.7 IC50 ChEMBL
O75716 STK16 Homo sapiens Human PF00069 7.7 pIC50 TTD_MultiTarget