Molecule Details
InChIKeyKFXHPWUOUVDXSQ-UHFFFAOYSA-N
Compound NameUS9790174, Example 10
Canonical SMILESCNc1cc(C(C)(C)C)cc(NC(=O)Nc2ccc(Oc3ccnc(Nc4cc(OC)cc(OCCOCCOCCOC)c4)n3)c(Cl)c2Cl)c1OC
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.07
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P12931 SRC Homo sapiens Human PF07714 PF00017 PF00018 7.7 IC50 ChEMBL;BindingDB
P43405 SYK Homo sapiens Human PF07714 PF00017 7.2 IC50 ChEMBL;BindingDB
Q16539 MAPK14 Homo sapiens Human PF00069 6.3 IC50 ChEMBL;BindingDB