Molecule Details
InChIKeyKFSJURQYNCYVKV-UHFFFAOYSA-N
Compound Name2-(dimethylamino)-N-[3-[[1-[2-(2-methylquinolin-5-yl)oxyethyl]piperidin-4-yl]methyl]phenyl]acetamide
Canonical SMILESCc1ccc2c(OCCN3CCC(Cc4cccc(NC(=O)CN(C)C)c4)CC3)cccc2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.33
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28221 HTR1D Homo sapiens Human PF00001 9.0 Ki ChEMBL;BindingDB
P28222 HTR1B Homo sapiens Human PF00001 8.2 Ki ChEMBL;BindingDB
P08908 HTR1A Homo sapiens Human PF00001 7.8 Ki ChEMBL;BindingDB