Molecule Details
InChIKeyKFRUZRAQPBNGME-UHFFFAOYSA-N
Compound NameN-[3-[3-[[6-(4-hydroxypiperidin-1-yl)-2-methylpyrimidin-4-yl]amino]-1H-pyrazol-5-yl]phenyl]benzenesulfonamide
Canonical SMILESCc1nc(Nc2cc(-c3cccc(NS(=O)(=O)c4ccccc4)c3)n[nH]2)cc(N2CCC(O)CC2)n1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.85
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P36888 FLT3 Homo sapiens Human PF00047 PF07714 8.0 IC50 ChEMBL;BindingDB
O14965 AURKA Homo sapiens Human PF00069 6.3 IC50 ChEMBL;BindingDB
Q02161 RHD Homo sapiens Human PF00909 6.3 pIC50 TTD_MultiTarget