Molecule Details
InChIKeyKEYFECUQJZMQPL-UHFFFAOYSA-N
Compound Name3-Amino-N-pyridin-3-yl-6-[4-(pyrrolidin-1-ylsulfonyl)phenyl]pyrazine-2-carboxamide
Canonical SMILESNc1ncc(-c2ccc(S(=O)(=O)N3CCCC3)cc2)nc1C(=O)Nc1cccnc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)4
Pfam Stratification Cross-Family
Avg pChEMBL7.02
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
P49841 GSK3B Homo sapiens Human PF00069 8.4 Ki ChEMBL;BindingDB
O96020 CCNE2 Homo sapiens Human PF02984 PF00134 6.6 Ki ChEMBL
P24864 CCNE1 Homo sapiens Human PF02984 PF00134 6.6 Ki ChEMBL
P24941 CDK2 Homo sapiens Human PF00069 6.6 Ki ChEMBL