Molecule Details
InChIKeyKEQSTBYHFUWBLB-UHFFFAOYSA-N
Compound Name3-[2-[2-Carbamoyl-6-(trifluoromethoxy)indol-1-yl]-4-pyridinyl]propanoic acid
Canonical SMILESNC(=O)c1cc2ccc(OC(F)(F)F)cc2n1-c1cc(CCC(=O)O)ccn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.42
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O15496 PLA2G10 Homo sapiens Human PF00068 6.6 IC50 ChEMBL;BindingDB
P14555 PLA2G2A Homo sapiens Human PF00068 6.5 IC50 ChEMBL;BindingDB
P39877 PLA2G5 Homo sapiens Human PF00068 6.1 IC50 ChEMBL;BindingDB