Molecule Details
InChIKeyKEPLBUUTAQCZOE-UHFFFAOYSA-N
Compound Name6-Ethyl-5-[3-(3-methoxy-5-pyridin-4-ylphenyl)but-1-ynyl]pyrimidine-2,4-diamine
Canonical SMILESCCc1nc(N)nc(N)c1C#CC(C)c1cc(OC)cc(-c2ccncc2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.23
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P0A017 folA Staphylococcus aureus Pathogen PF00186 7.7 Ki ChEMBL
P22906 DFR1 Candida albicans Pathogen PF00186 7.2 IC50 ChEMBL
J7IFZ2 Streptococcus pyogenes Pathogen PF00186 6.8 IC50 ChEMBL