Molecule Details
InChIKeyKEKBXAIGQLGOOL-UHFFFAOYSA-N
Compound Name7-[1-methyl-3-(trifluoromethyl)pyrazol-4-yl]-8,9,10,11-tetrahydro-3H-pyrazolo[4,3-a]phenanthridine
Canonical SMILESCn1cc(-c2nc3ccc4[nH]ncc4c3c3c2CCCC3)c(C(F)(F)F)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.25
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P36888 FLT3 Homo sapiens Human PF00047 PF07714 6.3 IC50 ChEMBL;BindingDB
P24941 CDK2 Homo sapiens Human PF00069 6.2 IC50 ChEMBL;BindingDB
P78396 CCNA1 Homo sapiens Human PF02984 PF00134 PF16500 6.2 IC50 ChEMBL