Molecule Details
InChIKeyKDCYOEAWXNGQEB-UHFFFAOYSA-N
Compound NameN-[4-[[4-[(5-methyl-1H-pyrazol-3-yl)amino]-6-morpholin-4-ylpyrimidin-2-yl]amino]phenyl]cyclopropanecarboxamide
Canonical SMILESCc1cc(Nc2cc(N3CCOCC3)nc(Nc3ccc(NC(=O)C4CC4)cc3)n2)n[nH]1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.41
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13546 RIPK1 Homo sapiens Human PF00531 PF07714 6.8 IC50 ChEMBL;BindingDB
O14965 AURKA Homo sapiens Human PF00069 6.4 IC50 ChEMBL;BindingDB
Q96GD4 AURKB Homo sapiens Human PF00069 6.1 IC50 ChEMBL;BindingDB