Molecule Details
InChIKeyKBWZVVPCJMAFMN-UHFFFAOYSA-N
Compound Name2-Amino-1-(3-hydroxy-2,6-dimethylphenyl)pyrrolo[3,2-b]quinoxaline-3-carboxamide
Canonical SMILESCc1ccc(O)c(C)c1-n1c(N)c(C(N)=O)c2nc3ccccc3nc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.16
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P54753 EPHB3 Homo sapiens Human PF14575 PF25599 PF01404 PF07699 PF00041 PF07714 PF00536 7.8 IC50 ChEMBL
Q99640 PKMYT1 Homo sapiens Human PF00069 7.5 IC50 ChEMBL
P30291 WEE1 Homo sapiens Human PF00069 6.2 IC50 ChEMBL