Molecule Details
InChIKeyKBKIOLUGZFJQBF-UHFFFAOYSA-N
Compound Name6-[1-[3-(2-methylquinolin-5-yl)oxypropyl]azetidin-3-yl]oxy-4H-1,4-benzoxazin-3-one
Canonical SMILESCc1ccc2c(OCCCN3CC(Oc4ccc5c(c4)NC(=O)CO5)C3)cccc2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.6
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08908 HTR1A Homo sapiens Human PF00001 6.8 Ki ChEMBL;BindingDB
P28221 HTR1D Homo sapiens Human PF00001 6.6 Ki ChEMBL;BindingDB
P28222 HTR1B Homo sapiens Human PF00001 6.4 Ki ChEMBL;BindingDB