Molecule Details
InChIKeyKBJSPAOJLUYMQM-UHFFFAOYSA-N
Compound NameN-(4-bromo-3-(1H-1,2,4-triazol-3-yl)thiophen-2-yl)-2-(6-cyano-2-oxoquinolin-1(2H)-yl)acetamide
Canonical SMILESN#Cc1ccc2c(ccc(=O)n2CC(=O)Nc2scc(Br)c2-c2ncn[nH]2)c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.57
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P45983 MAPK8 Homo sapiens Human PF00069 9.0 IC50 ChEMBL;BindingDB
P53779 MAPK10 Homo sapiens Human PF00069 8.7 IC50 ChEMBL;BindingDB
P45984 MAPK9 Homo sapiens Human PF00069 8.0 IC50 ChEMBL;BindingDB