Molecule Details
InChIKeyKAPNJGZVRYPTJW-UHFFFAOYSA-N
Compound Name5-[4-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-but-1-ynyl]-pyridin-2-ylamine
Canonical SMILESNc1ccc(C#CCCN2CC=C(c3ccccc3)CC2)cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.36
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P35462 DRD3 Homo sapiens Human PF00001 8.2 Ki ChEMBL;BindingDB
P21917 DRD4 Homo sapiens Human PF00001 6.6 Ki ChEMBL;BindingDB