Molecule Details
InChIKeyKAJHXHOIEARPHN-IRXDYDNUSA-N
Compound Name(6S,7S)-6-(4-m-tolyl-piperazine-1-carbonyl)-5-aza-spiro[2.5]octane-7-carboxylic acid hydroxyamide
Canonical SMILESCc1cccc(N2CCN(C(=O)[C@H]3NCC4(CC4)C[C@@H]3C(=O)NO)CC2)c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL6.97
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P08253 MMP2 Homo sapiens Human PF00040 PF00045 PF00413 7.2 pIC50 TTD_MultiTarget
O14672 ADAM10 Homo sapiens Human PF21299 PF00200 PF13574 6.7 IC50 ChEMBL;BindingDB