Molecule Details
InChIKeyKAHHZLXTLVPZAC-PKNBQFBNSA-N
Compound Name2-(2,5-dimethoxyphenyl)-N-(6-methyl-3-styryl-1H-indazol-5-yl)acetamide
Canonical SMILESCOc1ccc(OC)c(CC(=O)Nc2cc3c(/C=C/c4ccccc4)n[nH]c3cc2C)c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.17
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O14965 AURKA Homo sapiens Human PF00069 7.4 IC50 ChEMBL;BindingDB
O75716 STK16 Homo sapiens Human PF00069 7.4 pIC50 TTD_MultiTarget
Q96GD4 AURKB Homo sapiens Human PF00069 6.7 IC50 ChEMBL;BindingDB