Molecule Details
InChIKeyKAEBPVNZHCYYSN-UHFFFAOYSA-N
Compound Name4-(4-(1H-indol-3-yl)pyrimidin-2-ylamino)-N-ethylpiperidine-1-carboxamide
Canonical SMILESCCNC(=O)N1CCC(Nc2nccc(-c3c[nH]c4ccccc34)n2)CC1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.96
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P24941 CDK2 Homo sapiens Human PF00069 7.1 pIC50 TTD_MultiTarget
P45983 MAPK8 Homo sapiens Human PF00069 7.1 IC50 ChEMBL;BindingDB
P45984 MAPK9 Homo sapiens Human PF00069 6.6 IC50 ChEMBL;BindingDB