Molecule Details
InChIKeyJZNXPJAWGWXJFX-UHFFFAOYSA-N
Compound NamePyrazoloquinazoline deriv., 32
Canonical SMILESCCCN(CCO)CCCOc1ccc2c(Nc3cc(CC(=O)Nc4cccc(F)c4F)[nH]n3)ncnc2c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.46
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O14965 AURKA Homo sapiens Human PF00069 6.5 Ki ChEMBL;BindingDB
O75716 STK16 Homo sapiens Human PF00069 6.5 pIC50 TTD_MultiTarget