Molecule Details
InChIKeyJZHJELVVVUSHHT-QMMMGPOBSA-N
Compound Name(S)-4-Carbamoyl-2-(4-chloro-3-sulfamoyl-benzoylamino)-butyric acid
Canonical SMILESNC(=O)CC[C@H](NC(=O)c1ccc(Cl)c(S(N)(=O)=O)c1)C(=O)O
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.55
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00915 CA1 Homo sapiens Human PF00194 6.6 Ki ChEMBL;BindingDB
P00918 CA2 Homo sapiens Human PF00194 6.5 Ki ChEMBL;BindingDB
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 6.5 pIC50 TTD_MultiTarget