Molecule Details
InChIKeyJYYUWMLSDGSJDK-DMOWINQSSA-N
Canonical SMILESCOc1ccc([C@H]2[C@H](C(=O)O)[C@@H](c3ccc4c(c3)OCO4)CN2CC(=O)NC(c2ccccc2C)c2ccccc2C)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.88
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P24530 EDNRB Homo sapiens Human PF00001 9.0 IC50 ChEMBL;BindingDB
P25101 EDNRA Homo sapiens Human PF00001 6.8 IC50 ChEMBL;BindingDB