Molecule Details
InChIKeyJYIUNVOCEFIUIU-GHMZBOCLSA-N
Canonical SMILESC=CC(=O)N[C@@H]1CN(c2nc(Nc3cn(C)nc3OC)c3ncn(C)c3n2)C[C@H]1F
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.16
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB16228
Drug NameMavelertinib
CAS Number1776112-90-3
Groups investigational
ATC Codes nan
DescriptionMavelertinib is under investigation in clinical trial NCT02349633 (Study for Patients With NSCLC EGFR Mutations (Del 19 or L858R +/- T790M)).

Cross-references: BindingDB: 50450870 CHEMBL3989970 ChemSpider: 49070873 ZINC: ZINC000231225813
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P21860 ERBB3 Homo sapiens Human PF00757 PF14843 PF07714 PF01030 8.4 IC50 ChEMBL;BindingDB
P00533 EGFR Homo sapiens Human PF00757 PF14843 PF07714 PF01030 PF21314 7.9 IC50 ChEMBL;BindingDB