Molecule Details
InChIKeyJYHQBYXSPOBQMT-UHFFFAOYSA-N
Compound Name4-[6-(1,3-Difluoropropan-2-yloxy)-3-[(3,4-dimethoxyphenyl)methyl]-2,4-dioxoquinazolin-1-yl]piperidine-1-carbaldehyde
Canonical SMILESCOc1ccc(Cn2c(=O)c3cc(OC(CF)CF)ccc3n(C3CCN(C=O)CC3)c2=O)cc1OC
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.22
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13946 PDE7A Homo sapiens Human PF00233 7.4 IC50 ChEMBL;BindingDB
Q9NP56 PDE7B Homo sapiens Human PF00233 7.4 IC50 ChEMBL
O60658 PDE8A Homo sapiens Human PF00989 PF08629 PF23198 PF00233 6.8 IC50 ChEMBL;BindingDB