Molecule Details
InChIKeyJYASJBDXOVFRBN-PSXMRANNSA-N
Canonical SMILESO=S(=O)(Nc1ncnc2cc(N3CCN(Cc4ccccc4-c4ccc(Cl)cc4)CC3)ccc12)c1ccc(N[C@H](CCN2CCOCC2)CSc2ccccc2)c(S(=O)(=O)C(F)(F)F)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.45
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q07817 BCL2L1 Homo sapiens Human PF00452 PF02180 7.8 IC50 ChEMBL;BindingDB
P10415 BCL2 Homo sapiens Human PF00452 PF02180 7.1 IC50 ChEMBL;BindingDB