Molecule Details
InChIKeyJXTWQUKZLNDKPN-VOTSOKGWSA-N
Compound Name4-chloro-6-[[(E)-3-(1-methyl-[1,3]thiazolo[3,2-a]benzimidazol-2-yl)-3-oxoprop-1-enyl]amino]benzene-1,3-disulfonamide
Canonical SMILESCc1c(C(=O)/C=C/Nc2cc(Cl)c(S(N)(=O)=O)cc2S(N)(=O)=O)sc2nc3ccccc3n12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.63
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O43570 CA12 Homo sapiens Human PF00194 8.2 Ki ChEMBL;BindingDB
Q16790 CA9 Homo sapiens Human PF00194 7.5 Ki ChEMBL;BindingDB
P00918 CA2 Homo sapiens Human PF00194 7.2 Ki ChEMBL;BindingDB