Molecule Details
InChIKeyJXMNWIWHMKVRKH-UHFFFAOYSA-N
Compound Name4-[[3-[(1-propan-2-ylpiperidine-4-carbonyl)amino]phenyl]methylimino]-6,8a-dihydro-3H-quinazoline-8-carboxamide
Canonical SMILESCC(C)N1CCC(C(=O)Nc2cccc(CNC3=NC=NC4C(C(N)=O)=CCC=C34)c2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.57
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96GD4 AURKB Homo sapiens Human PF00069 8.7 IC50 ChEMBL;BindingDB
O14965 AURKA Homo sapiens Human PF00069 7.5 IC50 ChEMBL;BindingDB
P23443 RPS6KB1 Homo sapiens Human PF00069 PF00433 6.5 IC50 ChEMBL;BindingDB