Molecule Details
InChIKeyJWZSSEWMVYKYKW-UHFFFAOYSA-N
Compound Name3-[(3-Benzamido-4-Fluoranyl-Phenyl)amino]-~{n}-(2-Morpholin-4-Ylethyl)-11-Oxidanylidene-5,6-Dihydrodibenzo[1,2-~{d}:1',2'-~{f}][7]annulene-9-Carboxamide
Canonical SMILESO=C(NCCN1CCOCC1)c1ccc2c(c1)C(=O)c1ccc(Nc3ccc(F)c(NC(=O)c4ccccc4)c3)cc1CC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.86
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q16539 MAPK14 Homo sapiens Human PF00069 8.4 IC50 ChEMBL;BindingDB
Q15759 MAPK11 Homo sapiens Human PF00069 7.8 IC50 ChEMBL
P01375 TNF Homo sapiens Human PF00229 7.4 IC50 ChEMBL