Molecule Details
InChIKeyJWKZKADFQDTDIU-YJBOKZPZSA-N
Compound Name1,3-Thiazolidin-3-Yl[(2s,4s)-4-{4-[2-(Trifluoromethyl)quinolin-4-Yl]piperazin-1-Yl}pyrrolidin-2-Yl]methanone
Canonical SMILESO=C([C@@H]1C[C@H](N2CCN(c3cc(C(F)(F)F)nc4ccccc34)CC2)CN1)N1CCSC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.85
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P27487 DPP4 Homo sapiens Human PF00930 PF00326 9.4 IC50 ChEMBL;BindingDB
Q6V1X1 DPP8 Homo sapiens Human PF19520 PF00930 PF00326 7.1 IC50 ChEMBL;BindingDB
Q86TI2 DPP9 Homo sapiens Human PF19520 PF00930 PF00326 7.0 IC50 ChEMBL;BindingDB