Molecule Details
InChIKeyJWICEQLMDWKZGQ-UHFFFAOYSA-N
Compound Name10-chloro-2-methoxy-11H-indolo[3,2-c]quinoline-6-carboxylic acid
Canonical SMILESCOc1ccc2nc(C(=O)O)c3c4cccc(Cl)c4[nH]c3c2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.04
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13627 DYRK1A Homo sapiens Human PF00069 7.4 IC50 ChEMBL;BindingDB
P50750 CDK9 Homo sapiens Human PF00069 6.7 IC50 ChEMBL;BindingDB