Molecule Details
InChIKeyJWEJSOFKTOSBBW-UHFFFAOYSA-N
Compound NameN-(2-fluoro-4-methoxyphenyl)-6-(1H-pyrrolo[2,3-b]pyridin-3-yl)quinazolin-4-amine
Canonical SMILESCOc1ccc(Nc2ncnc3ccc(-c4c[nH]c5ncccc45)cc23)c(F)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)4
Pfam Stratification Cross-Family
Avg pChEMBL7.83
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13627 DYRK1A Homo sapiens Human PF00069 9.5 IC50 ChEMBL
P49841 GSK3B Homo sapiens Human PF00069 7.3 IC50 ChEMBL
O60563 CCNT1 Homo sapiens Human PF00134 PF21797 7.3 IC50 ChEMBL
P50750 CDK9 Homo sapiens Human PF00069 7.3 IC50 ChEMBL