Molecule Details
InChIKeyJWDZDXFXHWMSGR-QGZVFWFLSA-N
Compound Name4-[(3-methoxyphenyl)methyl]-2-[[(2R)-1-methylpyrrolidin-2-yl]methyl]phthalazin-1-one
Canonical SMILESCOc1cccc(Cc2nn(C[C@H]3CCCN3C)c(=O)c3ccccc23)c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.87
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35348 ADRA1A Homo sapiens Human PF00001 8.7 pIC50 TTD_MultiTarget
P35367 HRH1 Homo sapiens Human PF00001 8.7 Ki ChEMBL;BindingDB
Q9Y5N1 HRH3 Homo sapiens Human PF00001 6.2 Ki ChEMBL