Molecule Details
InChIKeyJVWOWDAKPHFJQW-HNNXBMFYSA-N
Compound Name6-(1-ethylpyrazol-4-yl)-1-[6-[(3S)-3-methylpiperazin-1-yl]-2-pyridinyl]pyrazolo[4,3-c]pyridine
Canonical SMILESCCn1cc(-c2cc3c(cn2)cnn3-c2cccc(N3CCN[C@@H](C)C3)n2)cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.02
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11309 PIM1 Homo sapiens Human PF00069 9.5 Ki ChEMBL;BindingDB
Q86V86 PIM3 Homo sapiens Human PF00069 9.5 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 8.1 Ki ChEMBL;BindingDB