Molecule Details
InChIKeyJVBGVXAXEZXWTE-MCUOQOIASA-N
Canonical SMILESCOc1cc(NC(=O)C[C@@]2(C)C[C@H](c3cccc(Cl)c3)[C@@H](c3ccc(Cl)cc3)N([C@H](CS(=O)(=O)C(C)(C)C)C3CC3)C2=O)ccc1C(=O)O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL9.95
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P08684 CYP3A4 Homo sapiens Human PF00067 10.3 IC50 ChEMBL;BindingDB
Q00987 MDM2 Homo sapiens Human PF02201 PF13920 PF00641 9.6 IC50 ChEMBL;BindingDB