Molecule Details
InChIKeyJVAUXOQNQAAUBJ-UHFFFAOYSA-N
Compound NameN-(6-(4-(3-(4-((5,6-dihydroimidazo[1,2-a]pyrazin-7(8H)-yl)methyl)-3-(trifluoromethyl)phenyl)ureido)phenoxy)pyrimidin-4-yl)cyclopropanecarboxamide
Canonical SMILESO=C(Nc1ccc(Oc2cc(NC(=O)C3CC3)ncn2)cc1)Nc1ccc(CN2CCn3ccnc3C2)c(C(F)(F)F)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.7
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P36888 FLT3 Homo sapiens Human PF00047 PF07714 8.5 IC50 ChEMBL;BindingDB
Q12866 MERTK Homo sapiens Human PF00041 PF00047 PF13927 PF07714 8.2 IC50 ChEMBL;BindingDB
P30530 AXL Homo sapiens Human PF00041 PF13927 PF07714 6.4 IC50 ChEMBL;BindingDB