Molecule Details
InChIKeyJUSJRQVEHUHMRQ-WOJBJXKFSA-N
Compound Name5-cyclopropyl-6-(2,6-dimethylpyridin-4-yl)-~{N}-[(3~{R},4~{R})-3-fluoranylpiperidin-4-yl]-1~{H}-indazol-3-amine
Canonical SMILESCc1cc(-c2cc3[nH]nc(N[C@@H]4CCNC[C@H]4F)c3cc2C2CC2)cc(C)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.95
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9NR97 TLR8 Homo sapiens Human PF13855 PF01582 9.2 IC50 ChEMBL;BindingDB
Q9NYK1 TLR7 Homo sapiens Human PF13855 PF01582 8.2 IC50 ChEMBL;BindingDB
Q9NR96 TLR9 Homo sapiens Human PF18837 PF13516 PF13855 PF01582 6.4 IC50 ChEMBL;BindingDB