Molecule Details
InChIKeyJUNKHWUBWMACDY-UHFFFAOYSA-N
Compound Name6-(4-chlorophenyl)-1-isopropyl-5-(4-methoxy-1-methyl-1H-benzo[d][1,2,3]triazol-6-yl)-2-(6-methoxypyridin-3-yl)-5,6-dihydropyrrolo[3,4-d]imidazol-4(1H)-one
Canonical SMILESCOc1ccc(-c2nc3c(n2C(C)C)C(c2ccc(Cl)cc2)N(c2cc(OC)c4nnn(C)c4c2)C3=O)cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.9
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P25440 BRD2 Homo sapiens Human PF17035 PF00439 7.0 IC50 ChEMBL;BindingDB
Q15059 BRD3 Homo sapiens Human PF17035 PF00439 7.0 IC50 ChEMBL;BindingDB
O60885 BRD4 Homo sapiens Human PF17035 PF17105 PF00439 6.7 IC50 ChEMBL;BindingDB