Molecule Details
InChIKeyJUMMJPACZXTMNS-HIFRSBDPSA-N
Compound Name(R)-3-amino-1-((S)-2-((6-(trifluoromethyl)pyridin-3-ylamino)methyl)pyrrolidin-1-yl)-4-(2,4,5-trifluorophenyl)butan-1-one
Canonical SMILESN[C@@H](CC(=O)N1CCC[C@H]1CNc1ccc(C(F)(F)F)nc1)Cc1cc(F)c(F)cc1F
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.85
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P27487 DPP4 Homo sapiens Human PF00930 PF00326 7.8 IC50 ChEMBL;BindingDB
Q86TI2 DPP9 Homo sapiens Human PF19520 PF00930 PF00326 6.5 IC50 ChEMBL;BindingDB
Q9UHL4 DPP7 Homo sapiens Human PF05577 6.3 IC50 ChEMBL;BindingDB