Molecule Details
InChIKeyJUKUQWGWZSESAV-UHFFFAOYSA-N
Compound NameN-(4-amino-5-chloro-6-ethoxypyridin-2-yl)-2-(4-methanesulfonyl-2,5-dimethoxyphenyl)acetamide
Canonical SMILESCCOc1nc(NC(=O)Cc2cc(OC)c(S(C)(=O)=O)cc2OC)cc(N)c1Cl
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.75
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P45983 MAPK8 Homo sapiens Human PF00069 8.1 Ki ChEMBL;BindingDB
P45984 MAPK9 Homo sapiens Human PF00069 7.9 Ki ChEMBL;BindingDB
P53779 MAPK10 Homo sapiens Human PF00069 7.2 Ki ChEMBL;BindingDB