Molecule Details
InChIKeyJUHFBGZNDZFVMC-UHFFFAOYSA-N
Compound Name4-(5-{[3-(3-Chloro-benzyl)-2-oxo-2,3,4,5-tetrahydro-1H-benzo[d]azepin-1-ylamino]-methyl}-imidazol-1-ylmethyl)-benzonitrile
Canonical SMILESN#Cc1ccc(Cn2cncc2CNC2C(=O)N(Cc3cccc(Cl)c3)CCc3ccccc32)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.64
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 7.6 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 7.6 IC50 ChEMBL