Molecule Details
InChIKeyJTVHPFGRRUKYMR-UHFFFAOYSA-N
Compound NameEthyl 4-cyano-2-(2-(4-methoxyphenyl)acetamido)thiophene-3-carboxylate
Canonical SMILESCCOC(=O)c1c(C#N)csc1NC(=O)Cc1ccc(OC)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.33
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P53779 MAPK10 Homo sapiens Human PF00069 6.5 IC50 ChEMBL;BindingDB
P45983 MAPK8 Homo sapiens Human PF00069 6.5 IC50 ChEMBL;BindingDB
P45984 MAPK9 Homo sapiens Human PF00069 6.0 IC50 ChEMBL;BindingDB